The leukotriene B4 receptor BLT1 is stabilized by transmembrane helix capping mutations
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Graphical abstract
Abbreviations
LTB4
leukotriene B4
GPCR
G-protein coupled receptor
gpBLT1
guinea pig leukotriene B4 receptor
TM helix
transmembrane helix
CPM
7-diethylamino-3-(4′-maleimidylphenyl)-4-methylcoumarin
Keywords
G-protein-coupled receptor
Leukotriene B4 receptor
Rational design mutation
Amino acid homology
Helix capping
Stabilization
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Copyright © 2015 The Authors. Published by Elsevier B.V.